|
Enantioselective binding of an acridine substituted Troeger s Base
to Calf Thymus DNA
Tatibouet,
Arnaud; Demeunynck, Martine; Lhomme, Jean; Dheu-Andries,
Marie-Louise; Charapoff, Denis; Vatton, Pierre;
Poster 022
Received: 22 Apr 1998
keywords: nitrogen heterocycle; acridine; Troeger's base; DNA
recognition DNA conformation;
|
 |
|
Synthesis of Modified Nucleosides by 1,3-Dipolar
Cycloaddition of C-Alcoxycarbonyl Nitrones
Chiacchio, Ugo;
Corsaro, Antonino; Gumina, Giuseppe; Rescifina, Antonio; Romeo,
Giovanni; Iannazzo, Daniela; Piperno, Anna;
Article 025
Received: 24 Apr 1998
keywords: 1,3-dipolar nitrone cycloaddition; isoxazolidines;
nucleoside analogues;
|
 |
|
Syntheses of New Cephalosporins as Potent Antibacterial
Agents
Hwu, Jih Ru; Tsay,
Shwu-Chen; Liao, Shu-Mei; Hakimelahi, Shahram;
Article 026
Received: 01 May 1998
keywords: Isodethiaazacephem; Mesylate; Triflate;
[1,4]-Elimination; Antibacterial; b-Lactam;
|
 |
|
A Novel Five-Step Route to the Synthesis of Psilocin from
Indole-3-carbaldehyde
Masanori Somei;
Fumio Yamada; Mayumi Tamura;
Poster 039
Received: 11 May 1998
keywords: psilocin; Indole-3-carbaldehyde;
4-Benzyloxyindole-3-carbaldehyde; 4-Benzyloxyindole-3-acetonitrile;
4-Benzyloxytryptamine;
|
 |
|
Strict Geometric Control in the Synthesis of
Porphyrin-Ligand Supramolecular Systems
Schultz, Austin C.;
Johnston, Martin R.; Warrener, Ronald N.; Gunter, Maxwell
J.;
Article 077
Received: 14 May 1998
keywords: cycloaddition; porphyrin; ligand; phenanthroline;
stereoselectivity;
|
 |
|
Synthesis and Antimicrobial Activity of Some
2-Alkyl-5,6-diphenylimidazo[2,1-b]thiazolidin-3-ones
Koos, Miroslav; Gajdos, Jan;
Steiner, Bohumil;
Poster 082
Received: 14 May 1998
keywords: Imidazo[2,1-b]thiazolidin-3-ones; antimicrobial
activity;
|
 |
|
Synthesis of Beta-carboline Derivatives and Their
Interaction with a DNA Oligomer
Konakahara, Takeo*;
Ozaki, Tomokazu; Komatsu, Harunobu; Ohta, Yuichi; Takeuchi, Hiroki;
Tamura, Sanae;
Poster 084
Received: 14 May 1998
keywords: DNA-intercalator; beta-carbolines; binding
constant; Scatchard plot; Synthesis;
|
 |
|
Synthesis of Novel Heterocyclic Systems from
a-(2-R-6-R1-5-halogenopyrimidin-4-yl)-2-azahetarylacetonitriles.
New Potential Anticancer Agents.
Fursy, Tamara;
Nemazany, Alexei; Rice, Kenner C.;
Poster 090
Received: 14 May 1998
keywords: condensed pyrimidines; new heterocyclic ring
systems; nucleophilic substitution; hetarylacetonitriles;
intermolecular cyclization; anticancer agents;
|
 |
|
Inhibition studies of Porphobilinogen Synthase from
Escherichia coli using diacids
Jarret, Caroline;
Bobalova, Janette; Stauffer, Frédéric; Henz,
Matthias; Neier, Reinhard;
Article 103
Received: 15 May 1998
keywords: Porphobilinogen; Porphobilinogen Synthase;
inhibition; diacids; 5-aminolevulinate; mechanism;
|
 |
|
Synthesis of 3-substituted analogues of levulinic acid via
Baylis-Hillman and Mukaiyama reactions. Potential inhibitors of
Porphobilinogen Synthase.
Bobál',
Pavel; Neier, Reinhard;
Article 104
Received: 15 May 1998
keywords: Porphobilinogen Synthase; levulinate; Mukaiyama;
Bailys-Hillman; Mitsunobu;
|
 |
|
Inhibition of porphobilinogen synthase (PBG-synthase) by
4,6-dioxoheptanoic acid (1) and related compounds
Stauffer,
Frédéric; Jarret, Caroline; Engeloch, Thomas; Henz,
Matthias; Bobalova, Janette; Neier, Reinhard;
Poster 107
Received: 15 May 1998
keywords: Porphobilinogen; porphobilinogen synthase;
inhibition; 1,3-diketone; 5-aminolevulinate;
|
 |
|
Regioselective bromination of the
16-hydroxymethyl-3-methoxyestra-1,3,5(10)-trien
isomers
Mernyák,
Erzsébet; Schneider, Gyula; Wölfling,
János;
Poster 115
Received: 15 May 1998
keywords: steroids; bromination; neighbouring group
participation;
|
 |
|
New pyrimidine cyclonucleosides with hydrogenated aglycone:
synthesis and structure
Shutalev, Anatoly D.; Gurskaya,
Galina V.;
Poster 116
Received: 15 May 1998
keywords: 2,3-O-isopropylideneribofuranosylamine;
isothiocyanatoaldehydes; pyrimidine cyclonucleosides;
3-(D-ribosyl)-4-hydroxyhexahydropyrimidine-2-thiones;
|
 |
|
Molecular imprinted polymers for the chiral separation of
pharmaceutically relevant heterocycles: First results of the
separation of the anti-Alzheimer drug Galanthamine
Jordis, Ulrich; Rizzi,
Andreas; Grohmann, Franz;
Poster 118
Received: 16 May 1998
keywords: Molecular imrinted polymers, MIP, chiral
separation, HPLC, CE, Galanthamine;
|
 |
Biologically Active Heterocycles/Target Oriented
Synthesis