The Cycle Formation
1. 5-Substituted Tetrazoles by 1,3-Dipolar Cycloaddition[1,2] |
|
2. 1,5-disubstituted tetrazoles by 1,3-dipolar cycloaddition [3] lgkR = r s I + lgko |
1.
t, oC | r | -lgko | |
80 | 3.35 | 5.99 | D # H = 50-60 kJ/mol |
90 | 3.37 | 5.69 | |
100 | 3.41 | 5.43 | D # S = -(120-200) J/mol K |
110 | 3.60 | 5.34 |
2.
t, oC | r | -lgko | |
60 | -0.94 | 7.43 | D # H = 85-90 kJ/mol |
80 | -1.08 | 6.64 | |
100 | - 0.99 | 5.84 | D # S = -(110-120) J/mol K |
1. I.E.Titova, V.S.Poplavskii, G.I. Koldobskii, V.A.Ostrovskii, Khim.Geterotsikl.Soedin., # 8, 1086-1089 (1986).
2.V.A.Ostrovskii,V.S.Poplavskii,G.I.Koldobskii,G.B.Erussalimsky,Khim.Geterotsikl.Soedin., # 9, 1214-1217 (1992).
3. A.A.Melnikov, M.M.Sokolova, M.A.Pervozvanskaja, V.V.Melnikov, Zh.Org.Khim., 15, # 9,1861-1866 (1979).