How does one describe the wavefunction for the π-complex formed from PhNHOPh?

January 25th, 2013

Although have dealt with the π-complex formed by protonation of PhNHOPh in several posts, there was one aspect that I had not really answered; what is the most appropriate description of its electronic nature? Here I do not so much provide an answer, as try to show how difficult getting an accurate answer might be.

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The demographics of a blog readership.

January 20th, 2013

With metrics in science publishing controversial to say the least, I pondered whether to write about the impact/influence a science-based blog might have (never mind whether it constitutes any measure of esteem). These are all terms that feature large when an (academic) organisation undertakes a survey of its researchers’ effectiveness. WordPress (the organisation that provides the software used for this blog) recently enhanced the stats it offers for its users, and one of these caught my eye.

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Aromaticity in the benzidine-like π-complex formed from PhNHOPh.

January 19th, 2013

The transient π-complex formed during the “[5,5]” sigmatropic rearrangement of protonated N,O-diphenyl hydroxylamine can be (formally) represented as below, namely the interaction of a six-π-electron aromatic ring (the phenoxide anion 2) with a four-π-electron phenyl dication-anion pair 1. Can one analyse this interaction in terms of aromaticity?

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The π-complex in the benzidine rearrangement: a molecular orbital analysis.

January 18th, 2013

Michael Dewar[cite]10.1016/S0040-4039(01)82765-9[/cite] famously implicated a so-called π-complex in the benzidine rearrangement, back in the days when quantum mechanical calculations could not yet provide a quantitatively accurate reality check. Because this π-complex actually remains a relatively unusual species to encounter in day-to-day chemistry, I thought I would try to show in a simple way how it forms.

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Why is N,O-diphenyl hydroxylamine (PhNHOPh) unknown?

January 16th, 2013

If you search e.g. Scifinder for N,O-diphenyl hydroxylamine (RN 24928-98-1) there is just one literature citation, to a 1962 patent. Nothing else; not even a calculation (an increasing proportion of the molecules reported in Chemical Abstracts have now only ever been subjected to calculation, not synthesis). A search of Reaxys also offers only one hit[cite]10.1016/S0040-4039(01)90757-9[/cite] reporting one unsuccessful attempt in 1963 to prepare this compound. Again, nothing else. Yet show this structure to most organic chemists, and I venture to suggest few would immediately predict this (unless they are experts on benzidine rearrangements).

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The strangely attractive conformation of C17H36.

January 13th, 2013

We tend to think of simple hydrocarbons as relatively inert and un-interesting molecules. However, a recent article[cite]10.1002/anie.201202894[/cite], which was in fact highlighted by Steve Bachrach on his blog , asks what “The Last Globally Stable Extended Alkane” might be. In other words, at what stage does a straight-chain hydrocarbon fold back upon itself, and no significant population of the linear form remain? The answer was suggested to be C17H36. I thought I might subject this conformation to an NCI (non-covalent-interaction) analysis.

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The Benzidine rearrangement. Computed kinetic isotope effects.

January 11th, 2013

Kinetic isotope effects have become something of a lost art when it comes to exploring reaction mechanisms. But in their heyday they were absolutely critical for establishing the mechanism of the benzidine rearrangement[cite]10.1021/ja00373a028[/cite]. This classic mechanism proceeds via bisprotonation of diphenyl hydrazine, but what happens next was the crux. Does this species rearrange directly to the C-C coupled intermediate (a concerted [5,5] sigmatropic reaction) or does it instead form a π-complex, as famously first suggested by Michael Dewar[cite]10.1016/S0040-4039(01)82765-9[/cite] [via TS(NN] and only then in a second step [via TS(CC)] form the C-C bond? Here I explore the isotope effects measured and calculated for this exact system.

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A conflation of concepts: Conformation and pericyclic.

January 10th, 2013

This is an interesting result I got when studying the [1,4] sigmatropic rearrangement of heptamethylbicyclo-[3.1.0]hexenyl cations. It fits into the last lecture of a series on pericyclic mechanisms, and just before the first lecture on conformational analysis. This is how they join.

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NCI (non-covalent-interaction) analysis for some π-hydrogen bonded systems.

January 8th, 2013

In this post, I looked at some hydrogen bonds formed by interaction of a π-system with an acidic hydrogen. Unlike normal lone pair donors, π-systems can involve more than two electrons, most commonly four or six. Here I look at examples of both these higher-order donors.

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Hidden intermediates in the benzidine rearrangement. The monoprotonated mechanism.

January 8th, 2013

Eagle-eyed footnote readers might have spotted one at the bottom of the post on the benzidine rearrangement. I was comparing the N-N bond lengths in crystal structures of known diprotonated hydrazines (~1.45Å) with the computed N-N bond length at the start point of the intrinsic reaction coordinate for the [5,5] sigmatropic rearrangement of di-N-protonated diphenylhydrazine (the active species in the benzidine rearrangement itself), which was some 1Å longer. This post explores the implications of this oddity.

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